eF-site ID 4qw5-I
PDB Code 4qw5
Chain I

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Title yCP beta5-M45A mutant in complex with carfilzomib
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Proteasome subunit alpha type-2
Source ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae;
Sequence I:  SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFE
KIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERA
IEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFI
AGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPE
DLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLK
MRQD
Description


Functional site

1) chain I
residue 124
type
sequence D
description BINDING SITE FOR RESIDUE 3BV H 301
source : AC3

2) chain I
residue 204
type
sequence D
description BINDING SITE FOR RESIDUE MG Y 302
source : BC6

3) chain I
residue 12-58
type prosite
sequence VAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLG
ITGLATD
description PROTEASOME_BETA_1 Proteasome beta-type subunits signature. LGIaGedFAVLAGDtrnitdysinsryep.KvfdcgdnivmsanGfaAD
source prosite : PS00854


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