|
eF-site ID
|
4qvy-L |
PDB Code
|
4qvy |
Chain
|
L |
|
click to enlarge
|
|
Title
|
yCP beta5-A49T-mutant in complex with bortezomib |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
PROTEASOME SUBUNIT ALPHA TYPE-2 |
Source
|
ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
L: |
QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYE
PKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHN
DKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKG
AVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQY
EPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGD
GLEILIVTKDGVRKEFYELKRD
|
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Description
|
|
Functional site
|
|
1)
|
chain |
L |
residue |
126 |
type |
|
sequence |
D
|
description |
BINDING SITE FOR RESIDUE BO2 K 301
|
source |
: AC6
|
|
2)
|
chain |
L |
residue |
222 |
type |
|
sequence |
D
|
description |
BINDING SITE FOR RESIDUE MG V 302
|
source |
: BC5
|
|
3)
|
chain |
L |
residue |
13-60 |
type |
prosite |
sequence |
LGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVM
SANGFAAD
|
description |
PROTEASOME_BETA_1 Proteasome beta-type subunits signature. VAMtGkdCVAIACDlrlgsqslgvsnkfe.Kifhyghvflgit.GlaTD
|
source |
prosite : PS00854
|
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