|
eF-site ID
|
4qh6-B |
PDB Code
|
4qh6 |
Chain
|
B |
|
click to enlarge
|
|
Title
|
Crystal structure of cruzain with nitrile inhibitor N-(2-AMINOETHYL)-NALPHA-BENZOYL-L-PHENYLALANINAMIDE |
Classification
|
Hydrolase/Hydrolase inhibitor |
Compound
|
Cruzipain |
Source
|
Trypanosoma cruzi (CYSP_TRYCR) |
|
Sequence
|
B: |
APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFL
AGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENN
GAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQ
DEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQL
DHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGS
NQCLVKEEASSAVVG
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
25 |
type |
ACT_SITE |
sequence |
C
|
description |
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
2)
|
chain |
B |
residue |
162 |
type |
ACT_SITE |
sequence |
H
|
description |
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
3)
|
chain |
B |
residue |
182 |
type |
ACT_SITE |
sequence |
N
|
description |
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
4)
|
chain |
B |
residue |
215 |
type |
SITE |
sequence |
G
|
description |
Cleavage; by autolysis => ECO:0000269|PubMed:1559982
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
5)
|
chain |
B |
residue |
47 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000255
|
source |
Swiss-Prot : SWS_FT_FI3
|
|
6)
|
chain |
B |
residue |
170 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000255
|
source |
Swiss-Prot : SWS_FT_FI3
|
|
|
|