eF-site ID 4pnk-B
PDB Code 4pnk
Chain B

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Title G protein-coupled receptor kinase 2 in complex with GSK180736A
Classification Transferase/Transferase inhibitor
Compound Beta-adrenergic receptor kinase 1
Source (GBG2_BOVIN)
Sequence B:  SELDQLRQEAEQLKNQIRDARKACADATLSQITNNIDPVG
RIQMRTRRTLRGHLAKIYAMHWGTDSRLLVSASQDGKLII
WDSYTTNKVHAIPLRSSWVMTCAYAPSGNYVACGGLDNIC
SIYNLKTREGNVRVSRELAGHTGYLSCCRFLDDNQIVTSS
GDTTCALWDIETGQQTTTFTGHTGDVMSLSLAPDTRLFVS
GACDASAKLWDVREGMCRQTFTGHESDINAICFFPNGNAF
ATGSDDATCRLFDLRADQELMTYSHDNIICGITSVSFSKS
GRLLLAGYDDFNCNVWDALKADRAGVLAGHDNRVSCLGVT
DDGMAVATGSWDSFLKIWN
Description


Functional site

1) chain B
residue 70-84
type prosite
sequence LVSASQDGKLIIWDS
description WD_REPEATS_1 Trp-Asp (WD) repeats signature. LVSAsqDgKLIIWDS
source prosite : PS00678

2) chain B
residue 157-171
type prosite
sequence IVTSSGDTTCALWDI
description WD_REPEATS_1 Trp-Asp (WD) repeats signature. LVSAsqDgKLIIWDS
source prosite : PS00678

3) chain B
residue 285-299
type prosite
sequence LLAGYDDFNCNVWDA
description WD_REPEATS_1 Trp-Asp (WD) repeats signature. LVSAsqDgKLIIWDS
source prosite : PS00678


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