eF-site ID 4pnk-A
PDB Code 4pnk
Chain A

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Title G protein-coupled receptor kinase 2 in complex with GSK180736A
Classification Transferase/Transferase inhibitor
Compound Beta-adrenergic receptor kinase 1
Source (GBG2_BOVIN)
Sequence A:  KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFR
DFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIF
DSYIMKELLACSHPFSKSATEHVQGHLGKKQVPPDLFQPY
IEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMN
DFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKM
KQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSF
ILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMH
NRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHA
SVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHS
PFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLL
QRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPP
LIPPREVNATKGIKLLDSDQELYRNFPLTISERWQQEVAE
TVFDTINAETDRLEARKKAKNKQLGHEEDYALGKDCIMHG
YMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTM
EEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQW
KKELRDAYREAQQLVQRVPKMKNKP
Description


Functional site

1) chain A
residue 197
type
sequence I
description binding site for residue KZQ A 701
source : AC1

2) chain A
residue 198
type
sequence G
description binding site for residue KZQ A 701
source : AC1

3) chain A
residue 199
type
sequence R
description binding site for residue KZQ A 701
source : AC1

4) chain A
residue 200
type
sequence G
description binding site for residue KZQ A 701
source : AC1

5) chain A
residue 205
type
sequence V
description binding site for residue KZQ A 701
source : AC1

6) chain A
residue 218
type
sequence A
description binding site for residue KZQ A 701
source : AC1

7) chain A
residue 222
type
sequence L
description binding site for residue KZQ A 701
source : AC1

8) chain A
residue 272
type
sequence D
description binding site for residue KZQ A 701
source : AC1

9) chain A
residue 274
type
sequence M
description binding site for residue KZQ A 701
source : AC1

10) chain A
residue 321
type
sequence A
description binding site for residue KZQ A 701
source : AC1

11) chain A
residue 322
type
sequence N
description binding site for residue KZQ A 701
source : AC1

12) chain A
residue 324
type
sequence L
description binding site for residue KZQ A 701
source : AC1

13) chain A
residue 334
type
sequence S
description binding site for residue KZQ A 701
source : AC1

14) chain A
residue 220
type MOD_RES
sequence K
description Cysteine methyl ester => ECO:0000269|PubMed:1903391
source Swiss-Prot : SWS_FT_FI2

15) chain A
residue 197-220
type prosite
sequence IGRGGFGEVYGCRKADTGKMYAMK
description PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGRGGFGEVYgCrkadtgkm..........YAMK
source prosite : PS00107

16) chain A
residue 313-325
type prosite
sequence VVYRDLKPANILL
description PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. VvYrDLKpaNILL
source prosite : PS00108


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