eF-site ID 4odf-A
PDB Code 4odf
Chain A

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Title Co-Crystal Structure of MDM2 with Inhibitor Compound 47
Classification LIGASE/LIGASE INHIBITOR
Compound E3 ubiquitin-protein ligase Mdm2
Source Homo sapiens (Human) (MDM2_HUMAN)
Sequence A:  GAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMK
EVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSF
SVKEHRKIYTMIYRNLVVV
Description


Functional site

1) chain A
residue 14
type
sequence V
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

2) chain A
residue 16
type
sequence T
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

3) chain A
residue 17
type
sequence S
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

4) chain A
residue 23
type
sequence E
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

5) chain A
residue 54
type
sequence L
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

6) chain A
residue 57
type
sequence L
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

7) chain A
residue 58
type
sequence G
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

8) chain A
residue 61
type
sequence I
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

9) chain A
residue 62
type
sequence M
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

10) chain A
residue 67
type
sequence Y
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

11) chain A
residue 93
type
sequence V
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

12) chain A
residue 96
type
sequence H
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

13) chain A
residue 99
type
sequence I
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

14) chain A
residue 100
type
sequence Y
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1

15) chain A
residue 104
type
sequence Y
description BINDING SITE FOR RESIDUE 2U1 A 201
source : AC1


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