eF-site ID 4oas-C
PDB Code 4oas
Chain C

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Title co-crystal structure of MDM2 (17-111) in complex with compound 25
Classification ligase/ligase inhibitor
Compound E3 ubiquitin-protein ligase Mdm2
Source Homo sapiens (Human) (MDM2_HUMAN)
Sequence C:  IPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLG
QYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRK
IYTMIYRNLVVV
Description


Functional site

1) chain C
residue 54
type
sequence L
description BINDING SITE FOR RESIDUE 2SW C 201
source : AC2

2) chain C
residue 58
type
sequence G
description BINDING SITE FOR RESIDUE 2SW C 201
source : AC2

3) chain C
residue 59
type
sequence Q
description BINDING SITE FOR RESIDUE 2SW C 201
source : AC2

4) chain C
residue 61
type
sequence I
description BINDING SITE FOR RESIDUE 2SW C 201
source : AC2

5) chain C
residue 93
type
sequence V
description BINDING SITE FOR RESIDUE 2SW C 201
source : AC2

6) chain C
residue 94
type
sequence K
description BINDING SITE FOR RESIDUE 2SW C 201
source : AC2

7) chain C
residue 96
type
sequence H
description BINDING SITE FOR RESIDUE 2SW C 201
source : AC2

8) chain C
residue 99
type
sequence I
description BINDING SITE FOR RESIDUE 2SW C 201
source : AC2

9) chain C
residue 51
type
sequence K
description BINDING SITE FOR RESIDUE SO4 E 202
source : AC4


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