eF-site ID 4jx7-B
PDB Code 4jx7
Chain B

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Title Crystal structure of Pim1 kinase in complex with inhibitor 2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6H)-one
Classification TRANSFERASE/TRANSFERASE INHIBITOR
Compound Serine/threonine-protein kinase pim-1
Source Homo sapiens (Human) (4JX7)
Sequence B:  KRRRH
Description


Functional site

1) chain B
residue 6
type
sequence R
description BINDING SITE FOR RESIDUE 1N6 A 401
source : AC1


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