|
eF-site ID
|
4jx7-B |
PDB Code
|
4jx7 |
Chain
|
B |
|
click to enlarge
|
|
Title
|
Crystal structure of Pim1 kinase in complex with inhibitor 2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6H)-one |
Classification
|
TRANSFERASE/TRANSFERASE INHIBITOR |
Compound
|
Serine/threonine-protein kinase pim-1 |
Source
|
Homo sapiens (Human) (4JX7) |
|
Sequence
|
B: |
KRRRH
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
6 |
type |
|
sequence |
R
|
description |
BINDING SITE FOR RESIDUE 1N6 A 401
|
source |
: AC1
|
|
|
|