eF-site ID 4hlm-A
PDB Code 4hlm
Chain A

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Title Crystal structure of Tankyrase 2 in complex with 3',4'-Dihydroxyflavone
Classification TRANSFERASE
Compound Tankyrase-2
Source (TNKS2_HUMAN)
Sequence A:  GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNR
YNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFH
GSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQY
VYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFS
A
Description


Functional site

1) chain A
residue 1081
type
sequence C
description BINDING SITE FOR RESIDUE ZN A 1201
source : AC1

2) chain A
residue 1084
type
sequence H
description BINDING SITE FOR RESIDUE ZN A 1201
source : AC1

3) chain A
residue 1089
type
sequence C
description BINDING SITE FOR RESIDUE ZN A 1201
source : AC1

4) chain A
residue 1092
type
sequence C
description BINDING SITE FOR RESIDUE ZN A 1201
source : AC1

5) chain A
residue 977
type
sequence R
description BINDING SITE FOR RESIDUE SO4 A 1202
source : AC2

6) chain A
residue 979
type
sequence H
description BINDING SITE FOR RESIDUE SO4 A 1202
source : AC2

7) chain A
residue 980
type
sequence R
description BINDING SITE FOR RESIDUE SO4 A 1202
source : AC2

8) chain A
residue 1067
type
sequence K
description BINDING SITE FOR RESIDUE SO4 A 1202
source : AC2

9) chain A
residue 1070
type
sequence Q
description BINDING SITE FOR RESIDUE SO4 A 1202
source : AC2

10) chain A
residue 990
type
sequence N
description BINDING SITE FOR RESIDUE SO4 A 1203
source : AC3

11) chain A
residue 991
type
sequence R
description BINDING SITE FOR RESIDUE SO4 A 1203
source : AC3

12) chain A
residue 1031
type
sequence H
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

13) chain A
residue 1032
type
sequence G
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

14) chain A
residue 1033
type
sequence S
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

15) chain A
residue 1050
type
sequence Y
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

16) chain A
residue 1060
type
sequence Y
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

17) chain A
residue 1067
type
sequence K
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

18) chain A
residue 1068
type
sequence S
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

19) chain A
residue 1071
type
sequence Y
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

20) chain A
residue 1075
type
sequence I
description BINDING SITE FOR RESIDUE 16S A 1204
source : AC4

21) chain A
residue 1081
type BINDING
sequence C
description BINDING => ECO:0000250|UniProtKB:O95271
source Swiss-Prot : SWS_FT_FI1

22) chain A
residue 1084
type BINDING
sequence H
description BINDING => ECO:0000250|UniProtKB:O95271
source Swiss-Prot : SWS_FT_FI1

23) chain A
residue 1089
type BINDING
sequence C
description BINDING => ECO:0000250|UniProtKB:O95271
source Swiss-Prot : SWS_FT_FI1

24) chain A
residue 1092
type BINDING
sequence C
description BINDING => ECO:0000250|UniProtKB:O95271
source Swiss-Prot : SWS_FT_FI1


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