eF-site ID 4gj8-B
PDB Code 4gj8
Chain B

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Title Crystal structure of renin in complex with PKF909-724 (compound 3)
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Renin
Source Homo sapiens (Human) (RENI_HUMAN)
Sequence B:  LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTG
SSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRY
STGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAE
FDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYN
RDSSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQM
KGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEA
LGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYV
FQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYT
EFDRRNNRIGFALAR
Description


Functional site

1) chain B
residue 32
type ACT_SITE
sequence D
description ACT_SITE => ECO:0000269|PubMed:20927107
source Swiss-Prot : SWS_FT_FI1

2) chain B
residue 215
type ACT_SITE
sequence D
description ACT_SITE => ECO:0000269|PubMed:20927107
source Swiss-Prot : SWS_FT_FI1

3) chain B
residue -1
type CARBOHYD
sequence N
description N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:2493678
source Swiss-Prot : SWS_FT_FI2

4) chain B
residue 67
type CARBOHYD
sequence N
description N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:2493678
source Swiss-Prot : SWS_FT_FI2


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