|
eF-site ID
|
4gj8-B |
PDB Code
|
4gj8 |
Chain
|
B |
|
click to enlarge
|
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Title
|
Crystal structure of renin in complex with PKF909-724 (compound 3) |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Renin |
Source
|
Homo sapiens (Human) (RENI_HUMAN) |
|
Sequence
|
B: |
LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTG
SSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRY
STGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAE
FDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYN
RDSSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQM
KGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEA
LGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYV
FQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYT
EFDRRNNRIGFALAR
|
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Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
32 |
type |
ACT_SITE |
sequence |
D
|
description |
ACT_SITE => ECO:0000269|PubMed:20927107
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
2)
|
chain |
B |
residue |
215 |
type |
ACT_SITE |
sequence |
D
|
description |
ACT_SITE => ECO:0000269|PubMed:20927107
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
3)
|
chain |
B |
residue |
-1 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:2493678
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
4)
|
chain |
B |
residue |
67 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:2493678
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
|
|