|
eF-site ID
|
4eu2-X |
PDB Code
|
4eu2 |
Chain
|
X |
|
click to enlarge
|
|
Title
|
Crystal structure of 20s proteasome with novel inhibitor K-7174 |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome component C7-alpha |
Source
|
ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
X: |
SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFE
KIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERA
IEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFI
AGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPE
DLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLK
MRQD
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
X |
residue |
61 |
type |
BINDING |
sequence |
K
|
description |
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
|
|