|
eF-site ID
|
4eu2-V |
PDB Code
|
4eu2 |
Chain
|
V |
|
click to enlarge
|
|
Title
|
Crystal structure of 20s proteasome with novel inhibitor K-7174 |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome component C7-alpha |
Source
|
ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
V: |
TSIMAVTFKDGVILGADSRTTTGAYIANRVTDKLTRVHDK
IWCCRSGSAADTQAIADIVQYHLELYTSQYGTPSTETAAS
VFKELCYENKDNLTAGIIVAGYDDKNKGEVYTIPLGGSVH
KLPYAIAGSGSTFIYGYCDKNFRENMSKEETVDFIKHSLS
QAIKWDGSSGGVIRMVVLTAAGVERLIFYPDEYEQL
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
V |
residue |
46 |
type |
|
sequence |
S
|
description |
BINDING SITE FOR RESIDUE WPI V 201
|
source |
: AC4
|
|
2)
|
chain |
V |
residue |
94 |
type |
|
sequence |
T
|
description |
BINDING SITE FOR RESIDUE WPI V 201
|
source |
: AC4
|
|
3)
|
chain |
V |
residue |
115 |
type |
|
sequence |
L
|
description |
BINDING SITE FOR RESIDUE WPI V 201
|
source |
: AC4
|
|
4)
|
chain |
V |
residue |
128 |
type |
|
sequence |
G
|
description |
BINDING SITE FOR RESIDUE WPI V 201
|
source |
: AC4
|
|
5)
|
chain |
V |
residue |
129 |
type |
|
sequence |
S
|
description |
BINDING SITE FOR RESIDUE WPI V 201
|
source |
: AC4
|
|
6)
|
chain |
V |
residue |
94 |
type |
|
sequence |
T
|
description |
BINDING SITE FOR RESIDUE WPI W 301
|
source |
: AC5
|
|
|
|