|
eF-site ID
|
4eu2-K |
PDB Code
|
4eu2 |
Chain
|
K |
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click to enlarge
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Title
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Crystal structure of 20s proteasome with novel inhibitor K-7174 |
Classification
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HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome component C7-alpha |
Source
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ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
K: |
MDIILGIRVQDSVILASSKAVTRGISVLKDSDDKTRQLSP
HTLMSFAGEAGDTVQFAEYIQANIQLYSIREDYELSPQAV
SSFVRQELAKSIRSRRPYQVNVLIGGYDKKKNKPELYQID
YLGTKVELPYGAHGYSGFYTFSLLDHHYRPDMTTEEGLDL
LKLCVQELEKRMPMDFKGVIVKIVDKDGIRQVDDFQ
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Description
|
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Functional site
|
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1)
|
chain |
K |
residue |
-1 |
type |
|
sequence |
M
|
description |
BINDING SITE FOR RESIDUE WPI L 301
|
source |
: AC3
|
|
2)
|
chain |
K |
residue |
22 |
type |
|
sequence |
R
|
description |
BINDING SITE FOR RESIDUE WPI L 301
|
source |
: AC3
|
|
3)
|
chain |
K |
residue |
23 |
type |
|
sequence |
G
|
description |
BINDING SITE FOR RESIDUE WPI L 301
|
source |
: AC3
|
|
4)
|
chain |
K |
residue |
4-51 |
type |
prosite |
sequence |
LGIRVQDSVILASSKAVTRGISVLKDSDDKTRQLSPHTLM
SFAGEAGD
|
description |
PROTEASOME_BETA_1 Proteasome beta-type subunits signature. VGVkGknCVVLGCErrstlklqdtritps.KvskidshvvlsfsGlnAD
|
source |
prosite : PS00854
|
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