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eF-site ID
|
4eu2-D |
PDB Code
|
4eu2 |
Chain
|
D |
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click to enlarge
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Title
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Crystal structure of 20s proteasome with novel inhibitor K-7174 |
Classification
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HYDROLASE/HYDROLASE INHIBITOR |
Compound
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Proteasome component C7-alpha |
Source
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ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
D: |
GYDRALSIFSPDGHIFQVEYALEAVKRGTCAVGVKGKNCV
VLGCERRSTLKLQDTRITPSKVSKIDSHVVLSFSGLNADS
RILIEKARVEAQSHRLTLEDPVTVEYLTRYVAGVQQRYTQ
SGGVRPFGVSTLIAGFDPRDDEPKLYQTEPSGIYSSWSAQ
TIGRNSKTVREFLEKNYDRKEPPATVEECVKLTVRSLLEV
VQTGAKNIEITVVKPDSDIVALSSEEINQYVTQIEQEKQE
Q
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Description
|
|
Functional site
|
|
1)
|
chain |
D |
residue |
4-26 |
type |
prosite |
sequence |
YDRALSIFSPDGHIFQVEYALEA
|
description |
PROTEASOME_ALPHA_1 Proteasome alpha-type subunits signature. YdralSiFSPdGHifQVEYAleA
|
source |
prosite : PS00388
|
|
2)
|
chain |
D |
residue |
34-81 |
type |
prosite |
sequence |
VGVKGKNCVVLGCERRSTLKLQDTRITPSKVSKIDSHVVL
SFSGLNAD
|
description |
PROTEASOME_BETA_1 Proteasome beta-type subunits signature. VGVkGknCVVLGCErrstlklqdtritps.KvskidshvvlsfsGlnAD
|
source |
prosite : PS00854
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