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eF-site ID
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4eu2-A |
PDB Code
|
4eu2 |
Chain
|
A |
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click to enlarge
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Title
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Crystal structure of 20s proteasome with novel inhibitor K-7174 |
Classification
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HYDROLASE/HYDROLASE INHIBITOR |
Compound
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Proteasome component C7-alpha |
Source
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ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
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Sequence
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A: |
AGYDRHITIFSPEGRLYQVEYAFKATNQTNINSLAVRGKD
CTVVISQKKVPDKLLDPTTVSYIFCISRTIGMVVNGPIPD
ARNAALRAKAEAAEFRYKYGYDMPCDVLAKRMANLSQIYT
QRAYMRPLGVILTFVSVDEELGPSIYKTDPAGYYVGYKAT
ATGPKQQEITTNLENHFKKSKIDHINEESWEKVVEFAITH
MIDALGTEFSKNDLEVGVATKDKFFTLSAENIEERLVAIA
E
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Description
|
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Functional site
|
|
1)
|
chain |
A |
residue |
12-34 |
type |
prosite |
sequence |
YDRHITIFSPEGRLYQVEYAFKA
|
description |
PROTEASOME_ALPHA_1 Proteasome alpha-type subunits signature. YdralSiFSPdGHifQVEYAleA
|
source |
prosite : PS00388
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