|
eF-site ID
|
4eu2-2 |
PDB Code
|
4eu2 |
Chain
|
2 |
|
click to enlarge
|
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Title
|
Crystal structure of 20s proteasome with novel inhibitor K-7174 |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome component C7-alpha |
Source
|
ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
2: |
TQQPIVTGTSVISMKYDNGVIIAADNLGSYGSLLRFNGVE
RLIPVGDNTVVGISGDISDMQHIERLLKDLVTENAYDNPL
ADAEEALEPSYIFEYLATVMYQRRSKMNPLWNAIIVAGVQ
SNGDQFLRYVNLLGVTYSSPTLATGFGAHMANPLLRKVVD
RESDIPKTTVQVAEEAIVNAMRVLYYRDARSSRNFSLAII
DKNTGLTFKKNLQVENMKWDFAKDIKGYGTQKI
|
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Description
|
|
Functional site
|
|
1)
|
chain |
2 |
residue |
-5 |
type |
|
sequence |
P
|
description |
BINDING SITE FOR RESIDUE WPI V 201
|
source |
: AC4
|
|
2)
|
chain |
2 |
residue |
-6 |
type |
|
sequence |
Q
|
description |
BINDING SITE FOR RESIDUE WPI V 201
|
source |
: AC4
|
|
3)
|
chain |
2 |
residue |
182 |
type |
|
sequence |
R
|
description |
BINDING SITE FOR RESIDUE WPI V 201
|
source |
: AC4
|
|
4)
|
chain |
2 |
residue |
4-51 |
type |
prosite |
sequence |
ISMKYDNGVIIAADNLGSYGSLLRFNGVERLIPVGDNTVV
GISGDISD
|
description |
PROTEASOME_BETA_1 Proteasome beta-type subunits signature. VGVkGknCVVLGCErrstlklqdtritps.KvskidshvvlsfsGlnAD
|
source |
prosite : PS00854
|
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