eF-site ID 4eop-D
PDB Code 4eop
Chain D

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Title Thr 160 phosphorylated CDK2 Q131E - human cyclin A3 complex with the inhibitor RO3306
Classification TRANSFERASE/TRANSFERASE INHIBITOR
Compound Cyclin-dependent kinase 2
Source Homo sapiens (Human) (CCNA2_HUMAN)
Sequence D:  VPDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRAIL
VDWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGKLQ
LVGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVLRM
EHLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESLAM
FLGELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSWPE
SLIRKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREKYK
NSKYHGVSLLNPPET
Description (1)  Cyclin-dependent kinase 2 (E.C.2.7.11.22), Cyclin-A2


Functional site

1) chain D
residue 200
type
sequence M
description BINDING SITE FOR RESIDUE MG D 501
source : AC4

2) chain D
residue 203
type
sequence Q
description BINDING SITE FOR RESIDUE MG D 501
source : AC4

3) chain D
residue 206
type
sequence I
description BINDING SITE FOR RESIDUE MG D 501
source : AC4


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