eF-site ID 4eok-B
PDB Code 4eok
Chain B

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Title Thr 160 phosphorylated CDK2 H84S, Q85M, K89D - human cyclin A3 complex with the inhibitor NU6102
Classification Transferase/Transferase Inhibitor
Compound Cyclin-dependent kinase 2
Source Homo sapiens (Human) (CCNA2_HUMAN)
Sequence B:  VPDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRAIL
VDWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGKLQ
LVGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVLRM
EHLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESLAM
FLGELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSWPE
SLIRKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREKYK
NSKYHGVSLLNPPETLNL
Description (1)  Cyclin-dependent kinase 2 (E.C.2.7.11.22), Cyclin-A2


Functional site

1) chain B
residue 189
type
sequence M
description BINDING SITE FOR RESIDUE SGM B 501
source : AC2

2) chain B
residue 193
type
sequence C
description BINDING SITE FOR RESIDUE SGM B 501
source : AC2

3) chain B
residue 211-242
type prosite
sequence RAILVDWLVEVGEEYKLQNETLHLAVNYIDRF
description CYCLINS Cyclins signature. RaiLvdWLvevgeeykLqnetLhlAVnYIDRF
source prosite : PS00292


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