|
eF-site ID
|
4eok-B |
PDB Code
|
4eok |
Chain
|
B |
|
click to enlarge
|
|
Title
|
Thr 160 phosphorylated CDK2 H84S, Q85M, K89D - human cyclin A3 complex with the inhibitor NU6102 |
Classification
|
Transferase/Transferase Inhibitor |
Compound
|
Cyclin-dependent kinase 2 |
Source
|
Homo sapiens (Human) (CCNA2_HUMAN) |
|
Sequence
|
B: |
VPDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRAIL
VDWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGKLQ
LVGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVLRM
EHLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESLAM
FLGELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSWPE
SLIRKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREKYK
NSKYHGVSLLNPPETLNL
|
|
Description
|
(1) |
Cyclin-dependent kinase 2 (E.C.2.7.11.22), Cyclin-A2
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
189 |
type |
|
sequence |
M
|
description |
BINDING SITE FOR RESIDUE SGM B 501
|
source |
: AC2
|
|
2)
|
chain |
B |
residue |
193 |
type |
|
sequence |
C
|
description |
BINDING SITE FOR RESIDUE SGM B 501
|
source |
: AC2
|
|
3)
|
chain |
B |
residue |
211-242 |
type |
prosite |
sequence |
RAILVDWLVEVGEEYKLQNETLHLAVNYIDRF
|
description |
CYCLINS Cyclins signature. RaiLvdWLvevgeeykLqnetLhlAVnYIDRF
|
source |
prosite : PS00292
|
|
|
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