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eF-site ID
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4cfx-D |
PDB Code
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4cfx |
Chain
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D |
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click to enlarge
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Title
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Structure-based design of C8-substituted O6-cyclohexylmethoxyguanine CDK1 and 2 inhibitors. |
Classification
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CELL CYCLE |
Compound
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CYCLIN-DEPENDENT KINASE 2 |
Source
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Homo sapiens (Human) (CCNA2_HUMAN) |
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Sequence
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D: |
NEVPDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRA
ILVDWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGK
LQLVGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVL
RMEHLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESL
AMFLGELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSW
PESLIRKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREK
YKNSKYHGVSLLNPPETLNL
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Description
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