|
eF-site ID
|
4cfx-B |
PDB Code
|
4cfx |
Chain
|
B |
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click to enlarge
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Title
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Structure-based design of C8-substituted O6-cyclohexylmethoxyguanine CDK1 and 2 inhibitors. |
Classification
|
CELL CYCLE |
Compound
|
CYCLIN-DEPENDENT KINASE 2 |
Source
|
Homo sapiens (Human) (CCNA2_HUMAN) |
|
Sequence
|
B: |
NEVPDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRA
ILVDWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGK
LQLVGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVL
RMEHLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESL
AMFLGELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSW
PESLIRKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREK
YKNSKYHGVSLLNPPETLNL
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Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
211-242 |
type |
prosite |
sequence |
RAILVDWLVEVGEEYKLQNETLHLAVNYIDRF
|
description |
CYCLINS Cyclins signature. RaiLvdWLvevgeeykLqnetLhlAVnYIDRF
|
source |
prosite : PS00292
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