|
eF-site ID
|
4cde-E |
PDB Code
|
4cde |
Chain
|
E |
|
click to enlarge
|
|
Title
|
Human DPP1 in complex with 4-amino-N-((1S)-1-cyano-2-(4-(4- cyanophenyl)phenyl)ethyl)tetrahydropyran-4-carboxamide |
Classification
|
HYDROLASE |
Compound
|
DIPEPTIDYL PEPTIDASE 1 EXCLUSION DOMAIN CHAIN |
Source
|
(CATC_HUMAN) |
|
Sequence
|
E: |
LPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEAR
IRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKY
AQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGG
FYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHH
T
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
E |
residue |
278 |
type |
ACT_SITE |
sequence |
F
|
description |
ACT_SITE => ECO:0000255|PROSITE-ProRule:PRU10090
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
2)
|
chain |
E |
residue |
280 |
type |
ACT_SITE |
sequence |
Y
|
description |
ACT_SITE => ECO:0000255|PROSITE-ProRule:PRU10090
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
3)
|
chain |
E |
residue |
323 |
type |
ACT_SITE |
sequence |
Y
|
description |
ACT_SITE => ECO:0000255|PROSITE-ProRule:PRU10090
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
4)
|
chain |
E |
residue |
252 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:19167329
|
source |
Swiss-Prot : SWS_FT_FI3
|
|
|
|