eF-site ID 4bv5-B PDB Code 4bv5 Chain B click to enlarge Title Identification of small molecule inhibitors selective for apo(a) kringles KIV-7, KIV-10 and KV. Classification HYDROLASE Compound APOLIPOPROTEIN(A) Source Homo sapiens (Human) (APOA_HUMAN) Sequence B:  CYHGNGQSYRGTFSTTVTGRTCQSWSSMTPHRHQRTPENY PNDGLTMNYCRNPDADTGPWCFTMDPSIRWEYCALTRC Description Functional site 1) chain B residue 67 type sequence D description BINDING SITE FOR RESIDUE 5C3 A 1081 source : AC1 2) chain B residue 68 type sequence P description BINDING SITE FOR RESIDUE 5C3 A 1081 source : AC1 3) chain B residue 69 type sequence S description BINDING SITE FOR RESIDUE 5C3 A 1081 source : AC1 4) chain B residue 33 type sequence H description BINDING SITE FOR RESIDUE 5C3 B 1081 source : AC2 5) chain B residue 34 type sequence Q description BINDING SITE FOR RESIDUE 5C3 B 1081 source : AC2 6) chain B residue 35 type sequence R description BINDING SITE FOR RESIDUE 5C3 B 1081 source : AC2 7) chain B residue 55 type sequence D description BINDING SITE FOR RESIDUE 5C3 B 1081 source : AC2 8) chain B residue 57 type sequence D description BINDING SITE FOR RESIDUE 5C3 B 1081 source : AC2 9) chain B residue 62 type sequence W description BINDING SITE FOR RESIDUE 5C3 B 1081 source : AC2 10) chain B residue 71 type sequence R description BINDING SITE FOR RESIDUE 5C3 B 1081 source : AC2 11) chain B residue 72 type sequence W description BINDING SITE FOR RESIDUE 5C3 B 1081 source : AC2

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