eF-site ID 4bv5-A
PDB Code 4bv5
Chain A

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Title Identification of small molecule inhibitors selective for apo(a) kringles KIV-7, KIV-10 and KV.
Classification HYDROLASE
Compound APOLIPOPROTEIN(A)
Source Homo sapiens (Human) (APOA_HUMAN)
Sequence A:  CYHGNGQSYRGTFSTTVTGRTCQSWSSMTPHRHQRTPENY
PNDGLTMNYCRNPDADTGPWCFTMDPSIRWEYCALTRC
Description


Functional site

1) chain A
residue 33
type
sequence H
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

2) chain A
residue 34
type
sequence Q
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

3) chain A
residue 35
type
sequence R
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

4) chain A
residue 55
type
sequence D
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

5) chain A
residue 57
type
sequence D
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

6) chain A
residue 62
type
sequence W
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

7) chain A
residue 64
type
sequence F
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

8) chain A
residue 71
type
sequence R
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

9) chain A
residue 72
type
sequence W
description BINDING SITE FOR RESIDUE 5C3 A 1081
source : AC1

10) chain A
residue 67
type
sequence D
description BINDING SITE FOR RESIDUE 5C3 B 1081
source : AC2

11) chain A
residue 68
type
sequence P
description BINDING SITE FOR RESIDUE 5C3 B 1081
source : AC2

12) chain A
residue 69
type
sequence S
description BINDING SITE FOR RESIDUE 5C3 B 1081
source : AC2

13) chain A
residue 50-63
type prosite
sequence YCRNPDADTGPWC
description KRINGLE_1 Kringle domain signature. YCRNpdadtgp.WC
source prosite : PS00021


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