eF-site ID 4bcn-B
PDB Code 4bcn
Chain B

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Title Structure of CDK2 in complex with cyclin A and a 2-amino-4-heteroaryl- pyrimidine inhibitor
Classification TRANSFERASE/CELL CYCLE
Compound CYCLIN-DEPENDENT KINASE 2
Source Homo sapiens (Human) (CCNA2_HUMAN)
Sequence B:  PDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRAILV
DWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGKLQL
VGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVLRME
HLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESLAMF
LGELSLIDADPYLKYLPSVIAAAAFHLALYTVTGQSWPES
LIRKTGYTLESLKPCLLDLHQTYLRAPKHAQQSIREKYKN
SKYHGVSLLNPPETLNL
Description (1)  CYCLIN-DEPENDENT KINASE 2 (E.C.2.7.11.22), CYCLIN-A2


Functional site

1) chain B
residue 199
type
sequence Y
description BINDING SITE FOR RESIDUE SO4 B 1433
source : AC3

2) chain B
residue 202
type
sequence K
description BINDING SITE FOR RESIDUE SO4 B 1433
source : AC3

3) chain B
residue 203
type
sequence Q
description BINDING SITE FOR RESIDUE SO4 B 1433
source : AC3

4) chain B
residue 243
type
sequence L
description BINDING SITE FOR RESIDUE SO4 B 1433
source : AC3

5) chain B
residue 245
type
sequence S
description BINDING SITE FOR RESIDUE SO4 B 1433
source : AC3

6) chain B
residue 246
type
sequence M
description BINDING SITE FOR RESIDUE SO4 B 1433
source : AC3

7) chain B
residue 247
type
sequence S
description BINDING SITE FOR RESIDUE SO4 B 1433
source : AC3

8) chain B
residue 211-242
type prosite
sequence RAILVDWLVEVGEEYKLQNETLHLAVNYIDRF
description CYCLINS Cyclins signature. RaiLvdWLvevgeeykLqnetLhlAVnYIDRF
source prosite : PS00292


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