eF-site ID 4aq3-C
PDB Code 4aq3
Chain C

click to enlarge
Title HUMAN BCL-2 WITH PHENYLACYLSULFONAMIDE INHIBITOR
Classification APOPTOSIS
Compound APOPTOSIS REGULATOR BCL-2, BCL-2-LIKE PROTEIN 1
Source Homo sapiens (Human) (BCLX_HUMAN)
Sequence C:  YDNREIVMKYIHYKLSQRGYEWDVVHLALRQAGDDFSRRY
RGDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIV
AFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTW
IQDNGGWDAFVELYG
Description (1)  APOPTOSIS REGULATOR BCL-2, BCL-2-LIKE PROTEIN 1


Functional site

1) chain C
residue 63
type
sequence F
description BINDING SITE FOR RESIDUE 398 C 1163
source : AC3

2) chain C
residue 67
type
sequence Y
description BINDING SITE FOR RESIDUE 398 C 1163
source : AC3

3) chain C
residue 70
type
sequence D
description BINDING SITE FOR RESIDUE 398 C 1163
source : AC3

4) chain C
residue 74
type
sequence M
description BINDING SITE FOR RESIDUE 398 C 1163
source : AC3

5) chain C
residue 95
type
sequence E
description BINDING SITE FOR RESIDUE 398 C 1163
source : AC3

6) chain C
residue 96
type
sequence L
description BINDING SITE FOR RESIDUE 398 C 1163
source : AC3

7) chain C
residue 161
type
sequence Y
description BINDING SITE FOR RESIDUE 398 C 1163
source : AC3

8) chain C
residue 58
type
sequence Q
description BINDING SITE FOR RESIDUE 398 F 1163
source : AC6

9) chain C
residue 160
type
sequence L
description BINDING SITE FOR RESIDUE 398 F 1163
source : AC6

10) chain C
residue 161
type
sequence Y
description BINDING SITE FOR RESIDUE 398 F 1163
source : AC6

11) chain C
residue 162
type
sequence G
description BINDING SITE FOR RESIDUE 398 F 1163
source : AC6

12) chain C
residue 72
type MOD_RES
sequence A
description Phosphoserine; by MAPK8 => ECO:0000269|PubMed:18570871
source Swiss-Prot : SWS_FT_FI4

13) chain C
residue 54
type MOD_RES
sequence L
description Phosphothreonine; by MAPK8 => ECO:0000269|PubMed:18570871
source Swiss-Prot : SWS_FT_FI2

14) chain C
residue 55
type MOD_RES
sequence A
description Phosphoserine; by MAPK8 and PKC => ECO:0000269|PubMed:18570871
source Swiss-Prot : SWS_FT_FI3


Display surface

Download
Links