eF-site ID 3wha-B
PDB Code 3wha
Chain B

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Title Hsp90 alpha N-terminal domain in complex with a tricyclic inhibitor
Classification Chaperone/chaperone Inhibitor
Compound Heat shock protein HSP 90-alpha
Source Homo sapiens (Human) (HS90A_HUMAN)
Sequence B:  EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDA
LDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTG
IGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFG
VGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTD
TGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIG
YPITLFVEK
Description


Functional site

1) chain B
residue 55
type
sequence A
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

2) chain B
residue 93
type
sequence D
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

3) chain B
residue 96
type
sequence I
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

4) chain B
residue 97
type
sequence G
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

5) chain B
residue 98
type
sequence M
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

6) chain B
residue 106
type
sequence N
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

7) chain B
residue 107
type
sequence L
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

8) chain B
residue 138
type
sequence F
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

9) chain B
residue 139
type
sequence Y
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

10) chain B
residue 184
type
sequence T
description BINDING SITE FOR RESIDUE WHA B 301
source : AC3

11) chain B
residue 51
type BINDING
sequence N
description
source Swiss-Prot : SWS_FT_FI1

12) chain B
residue 93
type BINDING
sequence D
description
source Swiss-Prot : SWS_FT_FI1

13) chain B
residue 138
type BINDING
sequence F
description
source Swiss-Prot : SWS_FT_FI1

14) chain B
residue 112
type BINDING
sequence K
description BINDING => ECO:0000250
source Swiss-Prot : SWS_FT_FI2

15) chain B
residue 58
type MOD_RES
sequence K
description N6-acetyllysine => ECO:0000250|UniProtKB:P07901
source Swiss-Prot : SWS_FT_FI3

16) chain B
residue 84
type MOD_RES
sequence K
description N6-acetyllysine => ECO:0000250|UniProtKB:P07901
source Swiss-Prot : SWS_FT_FI3


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