|
eF-site ID
|
3uzs-A |
PDB Code
|
3uzs |
Chain
|
A |
|
click to enlarge
|
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Title
|
Structure of the C13.28 RNA Aptamer Bound to the G Protein-Coupled Receptor Kinase 2-Heterotrimeric G Protein Beta 1 and Gamma 2 Subunit Complex |
Classification
|
TRANSFERASE/RNA |
Compound
|
Beta-adrenergic receptor kinase 1 |
Source
|
null (3UZS) |
|
Sequence
|
A: |
SKKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLF
RDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREI
FDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQP
YIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTM
NDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIK
MKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLS
FILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHM
HNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPH
ASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGH
SPVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVK
ESPFFRSLDWQMVFLQKYPPPLIPPRGEEDTKGIKLLDSD
QELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKT
KNKQLGHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFY
LFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLL
KIRGGKQFVLQCDSDPELVQWKKELRDAYREAQQLVQRVP
KMKNKPRAP
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Description
|
|
Functional site
|
|
1)
|
chain |
A |
residue |
335 |
type |
|
sequence |
D
|
description |
BINDING SITE FOR RESIDUE MG A 701
|
source |
: AC1
|
|
2)
|
chain |
A |
residue |
220 |
type |
MOD_RES |
sequence |
K
|
description |
Phosphohistidine => ECO:0000269|PubMed:12486123
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
3)
|
chain |
A |
residue |
670 |
type |
MOD_RES |
sequence |
A
|
description |
Phosphoserine => ECO:0000250|UniProtKB:P25098
|
source |
Swiss-Prot : SWS_FT_FI4
|
|
4)
|
chain |
A |
residue |
197-220 |
type |
prosite |
sequence |
IGRGGFGEVYGCRKADTGKMYAMK
|
description |
PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGRGGFGEVYgCrkadtgkm..........YAMK
|
source |
prosite : PS00107
|
|
5)
|
chain |
A |
residue |
313-325 |
type |
prosite |
sequence |
VVYRDLKPANILL
|
description |
PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. VvYrDLKpaNILL
|
source |
prosite : PS00108
|
|
|
|