eF-site ID 3tk6-A
PDB Code 3tk6
Chain A

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Title factor Xa in complex with D46-5241
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Factor X heavy chain
Source ORGANISM_COMMON: HUMAN; ORGANISM_SCIENTIFIC: Homo sapiens;
Sequence A:  IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTA
AHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRF
TKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLM
TQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSS
SFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVT
GIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK
Description (1)  Factor X heavy chain (E.C.3.4.21.6), Factor X light chain (E.C.3.4.21.6)


Functional site

1) chain A
residue 185
type
sequence Y
description BINDING SITE FOR RESIDUE CA A 261
source : AC1

2) chain A
residue 185
type
sequence Y
description BINDING SITE FOR RESIDUE CA A 261
source : AC1

3) chain A
residue 222
type
sequence R
description BINDING SITE FOR RESIDUE CA A 261
source : AC1

4) chain A
residue 224
type
sequence K
description BINDING SITE FOR RESIDUE CA A 261
source : AC1

5) chain A
residue 70
type
sequence D
description BINDING SITE FOR RESIDUE CA A 262
source : AC2

6) chain A
residue 72
type
sequence N
description BINDING SITE FOR RESIDUE CA A 262
source : AC2

7) chain A
residue 75
type
sequence Q
description BINDING SITE FOR RESIDUE CA A 262
source : AC2

8) chain A
residue 80
type
sequence E
description BINDING SITE FOR RESIDUE CA A 262
source : AC2

9) chain A
residue 97
type
sequence E
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

10) chain A
residue 98
type
sequence T
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

11) chain A
residue 99
type
sequence Y
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

12) chain A
residue 147
type
sequence E
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

13) chain A
residue 174
type
sequence F
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

14) chain A
residue 189
type
sequence D
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

15) chain A
residue 190
type
sequence A
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

16) chain A
residue 213
type
sequence V
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

17) chain A
residue 215
type
sequence W
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

18) chain A
residue 216
type
sequence G
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

19) chain A
residue 217
type
sequence E
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

20) chain A
residue 218
type
sequence G
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

21) chain A
residue 220
type
sequence C
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

22) chain A
residue 226
type
sequence G
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

23) chain A
residue 227
type
sequence I
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

24) chain A
residue 228
type
sequence Y
description BINDING SITE FOR RESIDUE D46 A 700
source : AC3

25) chain A
residue 57
type ACT_SITE
sequence H
description Charge relay system
source Swiss-Prot : SWS_FT_FI1

26) chain A
residue 102
type ACT_SITE
sequence D
description Charge relay system
source Swiss-Prot : SWS_FT_FI1

27) chain A
residue 195
type ACT_SITE
sequence S
description Charge relay system
source Swiss-Prot : SWS_FT_FI1

28) chain A
residue 53-58
type prosite
sequence LTAAHC
description TRYPSIN_HIS Serine proteases, trypsin family, histidine active site. LTAAHC
source prosite : PS00134

29) chain A
residue 189-200
type prosite
sequence DACQGDSGGPHV
description TRYPSIN_SER Serine proteases, trypsin family, serine active site. DAcqGDSGGPHV
source prosite : PS00135


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