|
eF-site ID
|
3shj-Z |
PDB Code
|
3shj |
Chain
|
Z |
|
click to enlarge
|
|
Title
|
Proteasome in complex with hydroxyurea derivative HU10 |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome component Y7 |
Source
|
ORGANISM_COMMON: yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
Z: |
QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYE
PKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHN
DKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKG
AVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQY
EPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGD
GLEILIVTKDGVRKEFYELKRD
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
Z |
residue |
112 |
type |
|
sequence |
S
|
description |
BINDING SITE FOR RESIDUE H10 Y 2I
|
source |
: AC4
|
|
2)
|
chain |
Z |
residue |
113 |
type |
|
sequence |
F
|
description |
BINDING SITE FOR RESIDUE H10 Y 2I
|
source |
: AC4
|
|
3)
|
chain |
Z |
residue |
118 |
type |
|
sequence |
S
|
description |
BINDING SITE FOR RESIDUE H10 Y 2I
|
source |
: AC4
|
|
4)
|
chain |
Z |
residue |
122 |
type |
|
sequence |
E
|
description |
BINDING SITE FOR RESIDUE H10 Y 2I
|
source |
: AC4
|
|
5)
|
chain |
Z |
residue |
125 |
type |
|
sequence |
R
|
description |
BINDING SITE FOR RESIDUE H10 Y 2I
|
source |
: AC4
|
|
|
|