eF-site ID 3r2a-D
PDB Code 3r2a
Chain D

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Title Crystal structure of RXRalpha ligand-binding domain complexed with corepressor SMRT2 and antagonist rhein
Classification TRANSCRIPTION
Compound Retinoic acid receptor RXR-alpha
Source Homo sapiens (Human) (NCOR2_HUMAN)
Sequence D:  NEDMPVERILEAELAVEPKTEPVTNICQAADKQLFTLVEW
AKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKD
GILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQM
DKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEA
YCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLI
GDTPIDTFLMEMLEAPHQM
Description


Functional site

1) chain D
residue 316
type BINDING
sequence R
description BINDING => ECO:0000269|PubMed:16107141, ECO:0000269|PubMed:18800767, ECO:0000269|PubMed:19167885, ECO:0007744|PDB:2ACL, ECO:0007744|PDB:3FAL, ECO:0007744|PDB:3FC6
source Swiss-Prot : SWS_FT_FI1

2) chain D
residue 327
type BINDING
sequence A
description BINDING => ECO:0000269|PubMed:16107141, ECO:0000269|PubMed:18800767, ECO:0000269|PubMed:19167885, ECO:0007744|PDB:2ACL, ECO:0007744|PDB:3FAL, ECO:0007744|PDB:3FC6
source Swiss-Prot : SWS_FT_FI1


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