eF-site ID 3psc-ABG
PDB Code 3psc
Chain A, B, G

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Title Bovine GRK2 in complex with Gbetagamma subunits
Classification TRANSFERASE/SIGNALING PROTEIN
Compound Beta-adrenergic receptor kinase 1
Source Bos taurus (Bovine) (GBG2_BOVIN)
Sequence A:  SKKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLF
RDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREI
FDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQP
YIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTM
NDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIK
MKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLS
FILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHM
HNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPH
ASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGH
SPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGL
LQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPP
PLIPPRGIKLLDSDQELYRNFPLTISERWQQEVAETVFDT
INAETDRLEARKKTKNKQLGHEEDYALGKDCIMHGYMSKM
GWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQI
KERKCLLLKIRGGKQFVLQCDSDPELVQWKKELRDAYREA
QQLVQRVPKMKNKP
B:  SELDQLRQEAEQLKNQIRDARKACADATLSQITNNIDPVG
RIQMRTRRTLRGHLAKIYAMHWGTDSRLLVSASQDGKLII
WDSYTTNKVHAIPLRSSWVMTCAYAPSGNYVACGGLDNIC
SIYNLKTREGNVRVSRELAGHTGYLSCCRFLDDNQIVTSS
GDTTCALWDIETGQQTTTFTGHTGDVMSLSLAPDTRLFVS
GACDASAKLWDVREGMCRQTFTGHESDINAICFFPNGNAF
ATGSDDATCRLFDLRADQELMTYSHDNIICGITSVSFSKS
GRLLLAGYDDFNCNVWDALKADRAGVLAGHDNRVSCLGVT
DDGMAVATGSWDSFLKIWN
G:  SIAQARKLVEQLKMEANIDRIKVSKAAADLMAYCEAHAKE
DPLLTPVPASENPFREKKFFX
Description


Functional site

1) chain G
residue 68
type MOD_RES
sequence X
description Cysteine methyl ester => ECO:0000269|PubMed:1903391
source Swiss-Prot : SWS_FT_FI2

2) chain A
residue 220
type MOD_RES
sequence K
description Cysteine methyl ester => ECO:0000269|PubMed:1903391
source Swiss-Prot : SWS_FT_FI2

3) chain G
residue 68
type LIPID
sequence X
description S-geranylgeranyl cysteine => ECO:0000269|PubMed:12764189, ECO:0000269|PubMed:1903391, ECO:0000269|PubMed:7626050
source Swiss-Prot : SWS_FT_FI3

4) chain B
residue 70-84
type prosite
sequence LVSASQDGKLIIWDS
description WD_REPEATS_1 Trp-Asp (WD) repeats signature. LVSAsqDgKLIIWDS
source prosite : PS00678

5) chain B
residue 157-171
type prosite
sequence IVTSSGDTTCALWDI
description WD_REPEATS_1 Trp-Asp (WD) repeats signature. LVSAsqDgKLIIWDS
source prosite : PS00678

6) chain B
residue 285-299
type prosite
sequence LLAGYDDFNCNVWDA
description WD_REPEATS_1 Trp-Asp (WD) repeats signature. LVSAsqDgKLIIWDS
source prosite : PS00678

7) chain A
residue 197-220
type prosite
sequence IGRGGFGEVYGCRKADTGKMYAMK
description PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGRGGFGEVYgCrkadtgkm..........YAMK
source prosite : PS00107

8) chain A
residue 313-325
type prosite
sequence VVYRDLKPANILL
description PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. VvYrDLKpaNILL
source prosite : PS00108


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