|
eF-site ID
|
3okj-Z |
PDB Code
|
3okj |
Chain
|
Z |
|
click to enlarge
|
|
Title
|
Alpha-keto-aldehyde binding mechanism reveals a novel lead structure motif for proteasome inhibition |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome component Y7 |
Source
|
ORGANISM_COMMON: yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
Z: |
QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYE
PKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHN
DKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKG
AVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQY
EPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGD
GLEILIVTKDGVRKEFYELKRD
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
Z |
residue |
114 |
type |
|
sequence |
D
|
description |
BINDING SITE FOR RESIDUE EP9 Y 300
|
source |
: AC2
|
|
2)
|
chain |
Z |
residue |
118 |
type |
|
sequence |
S
|
description |
BINDING SITE FOR RESIDUE EP9 Y 300
|
source |
: AC2
|
|
|
|