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eF-site ID
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3okj-W |
PDB Code
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3okj |
Chain
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W |
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click to enlarge
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Title
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Alpha-keto-aldehyde binding mechanism reveals a novel lead structure motif for proteasome inhibition |
Classification
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HYDROLASE/HYDROLASE INHIBITOR |
Compound
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Proteasome component Y7 |
Source
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ORGANISM_COMMON: yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
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Sequence
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W: |
SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFE
KIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERA
IEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFI
AGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPE
DLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLK
MRQD
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Description
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Functional site
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|
1)
|
chain |
W |
residue |
62 |
type |
BINDING |
sequence |
K
|
description |
|
source |
Swiss-Prot : SWS_FT_FI2
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