eF-site ID 3mu6-A
PDB Code 3mu6
Chain A

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Title Inhibiting the Binding of Class IIa Histone Deacetylases to Myocyte Enhancer Factor-2 by Small Molecules
Classification DNA BINDING PROTEIN/DNA
Compound Myocyte-specific enhancer factor 2A
Source Homo sapiens (Human) (3MU6)
Sequence A:  GRKKIQITRIMDERNRQVTFTKRKFGLMKKAYELSVLCDC
EIALIIFNSSNKLFQYASTDMDKVLLKYTAY
Description


Functional site

1) chain A
residue 61
type
sequence D
description BINDING SITE FOR RESIDUE BXL A 100
source : AC1

2) chain A
residue 62
type
sequence M
description BINDING SITE FOR RESIDUE BXL A 100
source : AC1

3) chain A
residue 63
type
sequence D
description BINDING SITE FOR RESIDUE BXL A 100
source : AC1

4) chain A
residue 66
type
sequence L
description BINDING SITE FOR RESIDUE BXL A 100
source : AC1

5) chain A
residue 67
type
sequence L
description BINDING SITE FOR RESIDUE BXL A 100
source : AC1

6) chain A
residue 70
type
sequence T
description BINDING SITE FOR RESIDUE BXL A 100
source : AC1

7) chain A
residue 59
type MOD_RES
sequence S
description Phosphoserine; by CK2 => ECO:0000250
source Swiss-Prot : SWS_FT_FI1

8) chain A
residue 3-57
type prosite
sequence RKKIQITRIMDERNRQVTFTKRKFGLMKKAYELSVLCDCE
IALIIFNSSNKLFQY
description MADS_BOX_1 MADS-box domain signature. RkKiqitrImDernRqvTFtKRKfgLmKKAyELSvLcdceIaLIIfnssnkLfqY
source prosite : PS00350


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