eF-site ID 3hvl-A
PDB Code 3hvl
Chain A

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Title Tethered PXR-LBD/SRC-1p complexed with SR-12813
Classification Transcription, Transferase
Compound Pregnane X receptor, Linker, Steroid receptor coactivator 1
Source Homo sapiens (Human) (NCOA1_HUMAN)
Sequence A:  GLTEEQRMMIRELMDAQMKTFDTTFSHFKNFRLPGVLSRE
EAAKWSQVRKDLCSLKVSLQLRGEDGSVWNYKPPADSGGK
EIFSLLPHMADMSTYMFKGIISFAKVISYFRDLPIEDQIS
LLKGAAFELCQLRFNTVFNAETGTWECGRLSYCLEQQLLL
EPMLKFHYMLKKLQLHEEEYVLMQAISLFSPDRPGVLQHR
VVDQLQEQFAITLKSYIECNRPQPAHRFLFLKIMAMLTEL
RSINAQHTQRLLRIQDIHPFATPLMQELFGITSLTERHKI
LHRLLQE
Description


Functional site

1) chain A
residue 243
type
sequence M
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

2) chain A
residue 246
type
sequence M
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

3) chain A
residue 247
type
sequence S
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

4) chain A
residue 251
type
sequence F
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

5) chain A
residue 281
type
sequence F
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

6) chain A
residue 285
type
sequence Q
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

7) chain A
residue 288
type
sequence F
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

8) chain A
residue 299
type
sequence W
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

9) chain A
residue 306
type
sequence Y
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

10) chain A
residue 323
type
sequence M
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

11) chain A
residue 407
type
sequence H
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

12) chain A
residue 411
type
sequence L
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

13) chain A
residue 420
type
sequence F
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

14) chain A
residue 425
type
sequence M
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

15) chain A
residue 429
type
sequence F
description BINDING SITE FOR RESIDUE SRL A 1
source : AC1

16) chain A
residue 247
type BINDING
sequence S
description BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
source Swiss-Prot : SWS_FT_FI1

17) chain A
residue 285
type BINDING
sequence Q
description BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
source Swiss-Prot : SWS_FT_FI1

18) chain A
residue 407
type BINDING
sequence H
description BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
source Swiss-Prot : SWS_FT_FI1


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