eF-site ID 3d36-ABC
PDB Code 3d36
Chain A, B, C

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Title How to Switch Off a Histidine Kinase: Crystal Structure of Geobacillus stearothermophilus KinB with the Inhibitor Sda
Classification Transferase/Transferase inhibitor
Compound Sporulation kinase B
Source (3D36)
Sequence A:  GPHMVIRLAASISHEIRNPLTAARGFIQLIEEQPLAADKR
RQYARIAIEELDRAEAIITDYLTFAKPAPETPEKLNVKLE
IERVIDILRPLANMSCVDIQATLAPFSVIGEREKFRQCLL
NVMKNAIEAMPNGGTLQVYVSIDNGRVLIRIADTGVGMTK
EQLERLGEPYFTTKGVKGTGLGMMVVYRIIESMNGTIRIE
SEIHKGTTVSIYLPLAS
B:  GPHMVIRAEKHLAASISHEIRNPLTAARGFIQLIEEQPLA
ADKRRQYARIAIEELDRAEAIITDYLTFAKPAPETPEKLN
VKLEIERVIDILRPLANMSCVDIQATLAPFSVIGEREKFR
QCLLNVMKNAIEAMPNGGTLQVYVSIDNGRVLIRIADTGV
GMTKEQLERLGEPYFTTKGVKGTGLGMMVVYRIIESMNGT
IRIESEIHKGTTVSIYLPLAS
C:  MKHLSDELLIESYFKAKELNLSPEFIELIEKEIQRRSLTH
KI
Description


Functional site

1) chain B
residue 324
type
sequence N
description BINDING SITE FOR RESIDUE MG B 477
source : AC1

2) chain A
residue 324
type
sequence N
description BINDING SITE FOR RESIDUE MG A 478
source : AC2

3) chain A
residue 324
type
sequence N
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

4) chain A
residue 328
type
sequence A
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

5) chain A
residue 352
type
sequence D
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

6) chain A
residue 356
type
sequence G
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

7) chain A
residue 357
type
sequence M
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

8) chain A
residue 365
type
sequence L
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

9) chain A
residue 370
type
sequence F
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

10) chain A
residue 371
type
sequence T
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

11) chain A
residue 372
type
sequence T
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

12) chain A
residue 373
type
sequence K
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

13) chain A
residue 377
type
sequence G
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

14) chain A
residue 378
type
sequence T
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

15) chain A
residue 379
type
sequence G
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

16) chain A
residue 380
type
sequence L
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

17) chain A
residue 381
type
sequence G
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

18) chain A
residue 382
type
sequence M
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

19) chain A
residue 406
type
sequence T
description BINDING SITE FOR RESIDUE ADP A 500
source : AC3

20) chain B
residue 324
type
sequence N
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

21) chain B
residue 328
type
sequence A
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

22) chain B
residue 352
type
sequence D
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

23) chain B
residue 356
type
sequence G
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

24) chain B
residue 357
type
sequence M
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

25) chain B
residue 365
type
sequence L
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

26) chain B
residue 370
type
sequence F
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

27) chain B
residue 371
type
sequence T
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

28) chain B
residue 372
type
sequence T
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

29) chain B
residue 373
type
sequence K
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

30) chain B
residue 378
type
sequence T
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

31) chain B
residue 379
type
sequence G
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

32) chain B
residue 380
type
sequence L
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

33) chain B
residue 381
type
sequence G
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

34) chain B
residue 382
type
sequence M
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

35) chain B
residue 406
type
sequence T
description BINDING SITE FOR RESIDUE ADP B 500
source : AC4

36) chain B
residue 224
type
sequence G
description BINDING SITE FOR RESIDUE MPD B 700
source : AC5

37) chain B
residue 225
type
sequence F
description BINDING SITE FOR RESIDUE MPD B 700
source : AC5

38) chain A
residue 237
type
sequence D
description BINDING SITE FOR RESIDUE MPD C 701
source : AC6

39) chain A
residue 238
type
sequence K
description BINDING SITE FOR RESIDUE MPD C 701
source : AC6

40) chain A
residue 241
type
sequence Q
description BINDING SITE FOR RESIDUE MPD C 701
source : AC6

41) chain B
residue 199
type
sequence E
description BINDING SITE FOR RESIDUE MPD C 701
source : AC6

42) chain B
residue 397
type
sequence R
description BINDING SITE FOR RESIDUE MPD C 701
source : AC6

43) chain B
residue 411
type
sequence Y
description BINDING SITE FOR RESIDUE MPD C 701
source : AC6

44) chain C
residue 5
type
sequence S
description BINDING SITE FOR RESIDUE MPD C 701
source : AC6

45) chain C
residue 8
type
sequence L
description BINDING SITE FOR RESIDUE MPD C 701
source : AC6

46) chain B
residue 211
type
sequence I
description BINDING SITE FOR RESIDUE MPD B 702
source : AC7

47) chain B
residue 260
type
sequence Y
description BINDING SITE FOR RESIDUE MPD B 702
source : AC7

48) chain A
residue 211
type
sequence I
description BINDING SITE FOR RESIDUE MPD B 703
source : AC8

49) chain A
residue 260
type
sequence Y
description BINDING SITE FOR RESIDUE MPD B 703
source : AC8

50) chain B
residue 266
type
sequence P
description BINDING SITE FOR RESIDUE MPD B 703
source : AC8


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