eF-site ID 3cdp-A
PDB Code 3cdp
Chain A

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Title Crystal structure of PPAR-gamma LBD complexed with a partial agonist, analogue of clofibric acid
Classification TRANSCRIPTION
Compound Peroxisome proliferator-activated receptor gamma
Source Homo sapiens (Human) (PPARG_HUMAN)
Sequence A:  ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSP
FVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQ
FRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEII
YTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEP
KFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPI
EDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIV
TEHVQLLQVIKKTETDMSLHPLLQEIYKDL
Description


Functional site

1) chain A
residue 282
type
sequence F
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

2) chain A
residue 285
type
sequence C
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

3) chain A
residue 286
type
sequence Q
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

4) chain A
residue 289
type
sequence S
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

5) chain A
residue 323
type
sequence H
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

6) chain A
residue 363
type
sequence F
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

7) chain A
residue 449
type
sequence H
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

8) chain A
residue 453
type
sequence L
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

9) chain A
residue 469
type
sequence L
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

10) chain A
residue 473
type
sequence Y
description BINDING SITE FOR RESIDUE YRG A 1
source : AC1

11) chain A
residue 286
type BINDING
sequence Q
description BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
source Swiss-Prot : SWS_FT_FI1

12) chain A
residue 323
type BINDING
sequence H
description BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
source Swiss-Prot : SWS_FT_FI1

13) chain A
residue 449
type BINDING
sequence H
description BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
source Swiss-Prot : SWS_FT_FI1

14) chain A
residue 473
type BINDING
sequence Y
description BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
source Swiss-Prot : SWS_FT_FI1


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