|
eF-site ID
|
3blr-B |
PDB Code
|
3blr |
Chain
|
B |
|
click to enlarge
|
|
Title
|
Crystal Structure of Human CDK9/cyclinT1 in complex with Flavopiridol |
Classification
|
TRANSCRIPTION |
Compound
|
Cell division protein kinase 9 |
Source
|
Homo sapiens (Human) (CCNT1_HUMAN) |
|
Sequence
|
B: |
NKRWYFTREQLENSPSRRFGVDPDKELSYRQQAANLLQDM
GQRLNVSQLTINTAIVYMHRFYMIQSFTRFPGNSVAPAAL
FLAAKVEGQPKKLEHVIKVAHTCLHPQESLPDTRSEAYLQ
QVQDLVILESIILQTLGFELTIDHPHTHVVKCTQLVRASK
DLAQTSYFMATNSLHLTTFSLQYTPPVVACVCIHLACKWS
NWEIPVSTDGKHWWEYVDATVTLELLDELTHELLQILEKT
PNRLKRIWNWR
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
99 |
type |
|
sequence |
K
|
description |
BINDING SITE FOR RESIDUE PO4 B 260
|
source |
: AC1
|
|
2)
|
chain |
B |
residue |
100 |
type |
|
sequence |
K
|
description |
BINDING SITE FOR RESIDUE PO4 B 260
|
source |
: AC1
|
|
3)
|
chain |
B |
residue |
103 |
type |
|
sequence |
H
|
description |
BINDING SITE FOR RESIDUE PO4 B 260
|
source |
: AC1
|
|
4)
|
chain |
B |
residue |
250 |
type |
|
sequence |
N
|
description |
BINDING SITE FOR RESIDUE PO4 B 261
|
source |
: AC3
|
|
5)
|
chain |
B |
residue |
254 |
type |
|
sequence |
R
|
description |
BINDING SITE FOR RESIDUE PO4 B 261
|
source |
: AC3
|
|
6)
|
chain |
B |
residue |
117 |
type |
MOD_RES |
sequence |
S
|
description |
Phosphoserine => ECO:0007744|PubMed:19369195
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
|
|