eF-site ID 3blr-B
PDB Code 3blr
Chain B

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Title Crystal Structure of Human CDK9/cyclinT1 in complex with Flavopiridol
Classification TRANSCRIPTION
Compound Cell division protein kinase 9
Source Homo sapiens (Human) (CCNT1_HUMAN)
Sequence B:  NKRWYFTREQLENSPSRRFGVDPDKELSYRQQAANLLQDM
GQRLNVSQLTINTAIVYMHRFYMIQSFTRFPGNSVAPAAL
FLAAKVEGQPKKLEHVIKVAHTCLHPQESLPDTRSEAYLQ
QVQDLVILESIILQTLGFELTIDHPHTHVVKCTQLVRASK
DLAQTSYFMATNSLHLTTFSLQYTPPVVACVCIHLACKWS
NWEIPVSTDGKHWWEYVDATVTLELLDELTHELLQILEKT
PNRLKRIWNWR
Description


Functional site

1) chain B
residue 99
type
sequence K
description BINDING SITE FOR RESIDUE PO4 B 260
source : AC1

2) chain B
residue 100
type
sequence K
description BINDING SITE FOR RESIDUE PO4 B 260
source : AC1

3) chain B
residue 103
type
sequence H
description BINDING SITE FOR RESIDUE PO4 B 260
source : AC1

4) chain B
residue 250
type
sequence N
description BINDING SITE FOR RESIDUE PO4 B 261
source : AC3

5) chain B
residue 254
type
sequence R
description BINDING SITE FOR RESIDUE PO4 B 261
source : AC3

6) chain B
residue 117
type MOD_RES
sequence S
description Phosphoserine => ECO:0007744|PubMed:19369195
source Swiss-Prot : SWS_FT_FI1


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