eF-site ID 2ycx-B
PDB Code 2ycx
Chain B

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Title TURKEY BETA1 ADRENERGIC RECEPTOR WITH STABILISING MUTATIONS AND BOUND ANTAGONIST CYANOPINDOLOL
Classification RECEPTOR
Compound BETA-1 ADRENERGIC RECEPTOR
Source (ADRB1_MELGA)
Sequence B:  QWEAGMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNL
FITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWT
SLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARA
KVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGC
CDFVTNRAYAIASSIISFYIPLLIMIFVALRVYREAKEQI
RKIDRASKRKRVMLMREHKALKTLGIIMGVFTLCWLPFFL
VNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPD
FRKAFKRLLA
Description


Functional site

1) chain B
residue 121
type BINDING
sequence D
description BINDING => ECO:0000269|PubMed:18594507, ECO:0007744|PDB:2VT4
source Swiss-Prot : SWS_FT_FI10

2) chain B
residue 211
type BINDING
sequence S
description BINDING => ECO:0000269|PubMed:18594507, ECO:0007744|PDB:2VT4
source Swiss-Prot : SWS_FT_FI10

3) chain B
residue 39-67
type TRANSMEM
sequence QWEAGMSLLMALVVLLIVAGNVLVIAAIG
description Helical; Name=1
source Swiss-Prot : SWS_FT_FI1

4) chain B
residue 77-103
type TRANSMEM
sequence NLFITSLACADLVVGLLVVPFGATLVV
description Helical; Name=2
source Swiss-Prot : SWS_FT_FI3

5) chain B
residue 116-137
type TRANSMEM
sequence LWTSLDVLCVTASIETLCVIAI
description Helical; Name=3
source Swiss-Prot : SWS_FT_FI5

6) chain B
residue 156-179
type TRANSMEM
sequence ARAKVIICTVWAISALVSFLPIMM
description Helical; Name=4
source Swiss-Prot : SWS_FT_FI6

7) chain B
residue 206-231
type TRANSMEM
sequence AYAIASSIISFYIPLLIMIFVALRVY
description Helical; Name=5
source Swiss-Prot : SWS_FT_FI7

8) chain B
residue 316-345
type TRANSMEM
sequence NRDLVPDWLFVAFNWLGYANSAMNPIIYCR
description Helical; Name=6
source Swiss-Prot : SWS_FT_FI8

9) chain B
residue 68-76
type TOPO_DOM
sequence STQRLQTLT
description Cytoplasmic => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI2

10) chain B
residue 138-155
type TOPO_DOM
sequence DRYLAITSPFRYQSLMTR
description Cytoplasmic => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI2

11) chain B
residue 232-315
type TOPO_DOM
sequence REAKEQIRKIDRASKRKRVMLMREHKALKTLGIIMGVFTL
CWLPFFLVNIVNVF
description Cytoplasmic => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI2

12) chain B
residue 104-115
type TOPO_DOM
sequence RGTWLWGSFLCE
description Extracellular => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI4

13) chain B
residue 180-205
type TOPO_DOM
sequence HWWRDEDPQALKCYQDPGCCDFVTNR
description Extracellular => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI4

14) chain B
residue 346-350
type TOPO_DOM
sequence SPDFR
description Extracellular => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI4


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