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eF-site ID
|
2y82-B |
PDB Code
|
2y82 |
Chain
|
B |
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click to enlarge
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Title
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Structure and property based design of factor Xa inhibitors: pyrrolidin-2-ones with aminoindane and phenylpyrrolidine P4 motifs |
Classification
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BLOOD CLOTTING |
Compound
|
ACTIVATED FACTOR XA HEAVY CHAIN |
Source
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ORGANISM_COMMON: HUMAN; ORGANISM_SCIENTIFIC: HOMO SAPIENS; |
|
Sequence
|
B: |
RKLCSLDNGDCDQFCHEEQNSVVCSCARGYTLADNGKACI
PTGPYPCGKQTLE
|
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Description
|
(1) |
ACTIVATED FACTOR XA HEAVY CHAIN (E.C.3.4.21.6), FACTOR X LIGHT CHAIN (E.C.3.4.21.6)
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Functional site
|
|
1)
|
chain |
B |
residue |
21-36 |
type |
prosite |
sequence |
CSCARGYTLADNGKAC
|
description |
EGF_2 EGF-like domain signature 2. CtCleGFegkn....C
|
source |
prosite : PS01186
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