eF-site ID 2xzd-A
PDB Code 2xzd
Chain A

click to enlarge
Title Caspase-3 in Complex with an Inhibitory DARPin-3.4
Classification HYDROLASE/PROTEIN BINDING
Compound CASPASE-3
Source Homo sapiens (Human) (2XZD)
Sequence A:  DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAAN
LRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSS
FVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTG
KPKLFIIQAXRGTELDCGIET
Description


Functional site

1) chain A
residue 51
type
sequence N
description BINDING SITE FOR RESIDUE MRD A 1175
source : AC1

2) chain A
residue 68
type
sequence D
description BINDING SITE FOR RESIDUE MRD A 1175
source : AC1

3) chain A
residue 71
type
sequence A
description BINDING SITE FOR RESIDUE MRD A 1175
source : AC1

4) chain A
residue 87
type
sequence N
description BINDING SITE FOR RESIDUE MRD A 1175
source : AC1

5) chain A
residue 89
type
sequence N
description BINDING SITE FOR RESIDUE MRD A 1175
source : AC1

6) chain A
residue 65
type
sequence S
description BINDING SITE FOR RESIDUE MPD B 1278
source : AC2

7) chain A
residue 107
type
sequence D
description BINDING SITE FOR RESIDUE MRD C 1177
source : AC4

8) chain A
residue 62
type catalytic
sequence T
description 815
source MCSA : MCSA1

9) chain A
residue 63
type catalytic
sequence S
description 815
source MCSA : MCSA1

10) chain A
residue 121
type catalytic
sequence H
description 815
source MCSA : MCSA1

11) chain A
residue 122
type catalytic
sequence G
description 815
source MCSA : MCSA1

12) chain A
residue 163
type catalytic
sequence X
description 815
source MCSA : MCSA1

13) chain A
residue 163
type MOD_RES
sequence X
description S-nitrosocysteine; in inhibited form => ECO:0000269|PubMed:10213689
source Swiss-Prot : SWS_FT_FI2

14) chain A
residue 108-122
type prosite
sequence HSKRSSFVCVLLSHG
description CASPASE_HIS Caspase family histidine active site. HskrsSfvCvLLSHG
source prosite : PS01121

15) chain A
residue 154-165
type prosite
sequence KPKLFIIQAXRG
description CASPASE_CYS Caspase family cysteine active site. KPKLFIIQACRG
source prosite : PS01122


Display surface

Download
Links