eF-site ID 2x9e-A
PDB Code 2x9e
Chain A

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Title HUMAN MPS1 IN COMPLEX WITH NMS-P715
Classification TRANSFERASE
Compound DUAL SPECIFICITY PROTEIN KINASE TTK
Source (TTK_HUMAN)
Sequence A:  NECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKY
VNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEIT
DQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEA
VHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANGTVNY
MPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQI
SKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRIS
IPELLAHPYVQIQT
Description


Functional site

1) chain A
residue 529
type
sequence K
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

2) chain A
residue 531
type
sequence I
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

3) chain A
residue 534
type
sequence G
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

4) chain A
residue 537
type
sequence S
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

5) chain A
residue 541
type
sequence Q
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

6) chain A
residue 551
type
sequence A
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

7) chain A
residue 553
type
sequence K
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

8) chain A
residue 586
type
sequence I
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

9) chain A
residue 603
type
sequence E
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

10) chain A
residue 604
type
sequence C
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

11) chain A
residue 605
type
sequence G
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

12) chain A
residue 606
type
sequence N
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

13) chain A
residue 607
type
sequence I
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

14) chain A
residue 611
type
sequence S
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

15) chain A
residue 652
type
sequence N
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

16) chain A
residue 654
type
sequence L
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

17) chain A
residue 663
type
sequence I
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

18) chain A
residue 664
type
sequence D
description BINDING SITE FOR RESIDUE SVE A 1796
source : AC1

19) chain A
residue 647
type ACT_SITE
sequence D
description Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00159, ECO:0000255|PROSITE-ProRule:PRU10027
source Swiss-Prot : SWS_FT_FI1

20) chain A
residue 531
type BINDING
sequence I
description BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
source Swiss-Prot : SWS_FT_FI2

21) chain A
residue 553
type BINDING
sequence K
description BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
source Swiss-Prot : SWS_FT_FI2

22) chain A
residue 531-553
type prosite
sequence IGSGGSSKVFQVLNEKKQIYAIK
description PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGSGGSSKVFqVlnekkqi...........YAIK
source prosite : PS00107

23) chain A
residue 643-655
type prosite
sequence IVHSDLKPANFLI
description PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. IvHsDLKpaNFLI
source prosite : PS00108


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