eF-site ID 2vvc-B
PDB Code 2vvc
Chain B

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Title Aminopyrrolidine Factor Xa inhibitor
Classification HYDROLASE
Compound ACTIVATED FACTOR XA HEAVY CHAIN
Source Homo sapiens (Human) (FA10_HUMAN)
Sequence B:  IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTA
AHCLYQAKRFKVRVGGGEAVHEVEVVIKHNRFTKETYDFD
IAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVS
GFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNM
FCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEG
CARKGKYGIYTKVTAFLKWIDRSMK
Description


Functional site

1) chain B
residue 97
type
sequence E
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

2) chain B
residue 98
type
sequence T
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

3) chain B
residue 147
type
sequence E
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

4) chain B
residue 174
type
sequence F
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

5) chain B
residue 189
type
sequence D
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

6) chain B
residue 190
type
sequence A
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

7) chain B
residue 192
type
sequence Q
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

8) chain B
residue 195
type
sequence S
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

9) chain B
residue 213
type
sequence V
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

10) chain B
residue 215
type
sequence W
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

11) chain B
residue 216
type
sequence G
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

12) chain B
residue 217
type
sequence E
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

13) chain B
residue 218
type
sequence G
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

14) chain B
residue 220
type
sequence C
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

15) chain B
residue 226
type
sequence G
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

16) chain B
residue 227
type
sequence I
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

17) chain B
residue 228
type
sequence Y
description BINDING SITE FOR RESIDUE LZF B 1244
source : AC2

18) chain B
residue 185
type
sequence Y
description BINDING SITE FOR RESIDUE NA B 1245
source : AC5

19) chain B
residue 185
type
sequence Y
description BINDING SITE FOR RESIDUE NA B 1245
source : AC5

20) chain B
residue 222
type
sequence R
description BINDING SITE FOR RESIDUE NA B 1245
source : AC5

21) chain B
residue 224
type
sequence K
description BINDING SITE FOR RESIDUE NA B 1245
source : AC5

22) chain B
residue 57
type ACT_SITE
sequence H
description Charge relay system
source Swiss-Prot : SWS_FT_FI1

23) chain B
residue 102
type ACT_SITE
sequence D
description Charge relay system
source Swiss-Prot : SWS_FT_FI1

24) chain B
residue 195
type ACT_SITE
sequence S
description Charge relay system
source Swiss-Prot : SWS_FT_FI1


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