eF-site ID 2vt4-A
PDB Code 2vt4
Chain A

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Title TURKEY BETA1 ADRENERGIC RECEPTOR WITH STABILISING MUTATIONS AND BOUND CYANOPINDOLOL
Classification RECEPTOR
Compound BETA1 ADRENERGIC RECEPTOR
Source (ADRB1_MELGA)
Sequence A:  WEAGMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLF
ITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTS
LDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAK
VIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCC
DFVTNRAYAIASSIISFYIPLLIMIFVALRVYREAKEQIR
EHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWL
FVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLLA
Description


Functional site

1) chain A
residue 68-76
type TOPO_DOM
sequence STQRLQTLT
description Cytoplasmic => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI2

2) chain A
residue 138-155
type TOPO_DOM
sequence DRYLAITSPFRYQSLMTR
description Cytoplasmic => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI2

3) chain A
residue 232-315
type TOPO_DOM
sequence REAKEQIREHKALKTLGIIMGVFTLCWLPFFLVNIVNVF
description Cytoplasmic => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI2

4) chain A
residue 104-115
type TOPO_DOM
sequence RGTWLWGSFLCE
description Extracellular => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI4

5) chain A
residue 180-205
type TOPO_DOM
sequence HWWRDEDPQALKCYQDPGCCDFVTNR
description Extracellular => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI4

6) chain A
residue 316-320
type TOPO_DOM
sequence NRDLV
description Extracellular => ECO:0000269|PubMed:18594507
source Swiss-Prot : SWS_FT_FI4

7) chain A
residue 121
type BINDING
sequence D
description BINDING => ECO:0000269|PubMed:18594507, ECO:0007744|PDB:2VT4
source Swiss-Prot : SWS_FT_FI10

8) chain A
residue 211
type BINDING
sequence S
description BINDING => ECO:0000269|PubMed:18594507, ECO:0007744|PDB:2VT4
source Swiss-Prot : SWS_FT_FI10

9) chain A
residue 329
type BINDING
sequence N
description BINDING => ECO:0000269|PubMed:18594507, ECO:0007744|PDB:2VT4
source Swiss-Prot : SWS_FT_FI10

10) chain A
residue 358
type LIPID
sequence A
description S-palmitoyl cysteine => ECO:0000250
source Swiss-Prot : SWS_FT_FI11

11) chain A
residue 127-143
type prosite
sequence ASIETLCVIAIDRYLAI
description G_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. ASIeTLCVIAIDRYLaI
source prosite : PS00237

12) chain A
residue 77-103
type TRANSMEM
sequence NLFITSLACADLVVGLLVVPFGATLVV
description Helical; Name=2
source Swiss-Prot : SWS_FT_FI3

13) chain A
residue 116-137
type TRANSMEM
sequence LWTSLDVLCVTASIETLCVIAI
description Helical; Name=3
source Swiss-Prot : SWS_FT_FI5

14) chain A
residue 156-179
type TRANSMEM
sequence ARAKVIICTVWAISALVSFLPIMM
description Helical; Name=4
source Swiss-Prot : SWS_FT_FI6

15) chain A
residue 206-231
type TRANSMEM
sequence AYAIASSIISFYIPLLIMIFVALRVY
description Helical; Name=5
source Swiss-Prot : SWS_FT_FI7

16) chain A
residue 286-315
type TRANSMEM
sequence HKALKTLGIIMGVFTLCWLPFFLVNIVNVF
description Helical; Name=6
source Swiss-Prot : SWS_FT_FI8

17) chain A
residue 321-343
type TRANSMEM
sequence PDWLFVAFNWLGYANSAMNPIIY
description Helical; Name=7
source Swiss-Prot : SWS_FT_FI9


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