eF-site ID 2vh0-B
PDB Code 2vh0
Chain B

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Title Structure and property based design of factor Xa inhibitors:biaryl pyrrolidin-2-ones incorporating basic heterocyclic motifs
Classification HYDROLASE
Compound ACTIVATED FACTOR XA HEAVY CHAIN
Source ORGANISM_COMMON: HUMAN; ORGANISM_SCIENTIFIC: HOMO SAPIENS;
Sequence B:  RKLCSLDNGDCDQFCHEEQNSVVCSCARGYTLADNGKACI
PTGPYPCGKQTL
Description (1)  ACTIVATED FACTOR XA HEAVY CHAIN (E.C.3.4.21.6), ACTIVATED FACTOR XA LIGHT CHAIN (E.C.3.4.21.6)


Functional site

1) chain B
residue 21-36
type prosite
sequence CSCARGYTLADNGKAC
description EGF_2 EGF-like domain signature 2. CtCleGFegkn....C
source prosite : PS01186


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