|
eF-site ID
|
2r0k-A |
PDB Code
|
2r0k |
Chain
|
A |
|
click to enlarge
|
|
Title
|
Protease domain of HGFA with inhibitor Fab58 |
Classification
|
HYDROLASE, IMMUNE SYSTEM |
Compound
|
Hepatocyte growth factor activator |
Source
|
Homo sapiens (Human) (2R0K) |
|
Sequence
|
A: |
IIGGSSSLPGSHPWLAAIYIGDSFCAGSLVHTCWVVSAAH
CFSHSPPRDSVSVVLGQHFFNRTTDVTQTFGIEKYIPYTL
YSVFNPSDHDLVLIRLKKKGDRCATRSQFVQPICLPEPGS
TFPAGHKCQIAGWGHLDENVSGYSSSLREALVPLVADHKC
SSPEVYGADISPNMLCAGYFDCKSDACQGDSGGPLACEKN
GVAYLYGIISWGDGCGRLHKPGVYTRVANYVDWINDRIR
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
A |
residue |
53-58 |
type |
prosite |
sequence |
VSAAHC
|
description |
TRYPSIN_HIS Serine proteases, trypsin family, histidine active site. VSAAHC
|
source |
prosite : PS00134
|
|
2)
|
chain |
A |
residue |
189-200 |
type |
prosite |
sequence |
DACQGDSGGPLA
|
description |
TRYPSIN_SER Serine proteases, trypsin family, serine active site. DAcqGDSGGPLA
|
source |
prosite : PS00135
|
|
3)
|
chain |
A |
residue |
57 |
type |
ACT_SITE |
sequence |
H
|
description |
Charge relay system => ECO:0000269|PubMed:15713485
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
4)
|
chain |
A |
residue |
102 |
type |
ACT_SITE |
sequence |
D
|
description |
Charge relay system => ECO:0000269|PubMed:15713485
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
5)
|
chain |
A |
residue |
195 |
type |
ACT_SITE |
sequence |
S
|
description |
Charge relay system => ECO:0000269|PubMed:15713485
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
6)
|
chain |
A |
residue |
74 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:16335952, ECO:0000269|PubMed:18077410, ECO:0000269|PubMed:19159218
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
7)
|
chain |
A |
residue |
147 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000255
|
source |
Swiss-Prot : SWS_FT_FI3
|
|
|
|