eF-site ID 2q5p-B
PDB Code 2q5p
Chain B

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Title Crystal Structure of PPARgamma bound to partial agonist MRL24
Classification Ligand binding protein
Compound Peroxisome Proliferator-Activated Receptor gamma
Source Homo sapiens (Human) (PPARG_HUMAN)
Sequence B:  ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKSPFVIY
DMNSLMMGEFKHITVAIRIFQGCQFRSVEAVQEITEYAKS
IPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLIS
EGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDS
DLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLK
LNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVILHPLLQ
EIYKD
Description


Functional site

1) chain B
residue 226
type
sequence F
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

2) chain B
residue 264
type
sequence F
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

3) chain B
residue 284
type
sequence G
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

4) chain B
residue 285
type
sequence C
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

5) chain B
residue 288
type
sequence R
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

6) chain B
residue 289
type
sequence S
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

7) chain B
residue 292
type
sequence A
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

8) chain B
residue 326
type
sequence I
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

9) chain B
residue 327
type
sequence Y
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

10) chain B
residue 329
type
sequence M
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

11) chain B
residue 330
type
sequence L
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

12) chain B
residue 333
type
sequence L
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

13) chain B
residue 340
type
sequence L
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

14) chain B
residue 341
type
sequence I
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

15) chain B
residue 342
type
sequence S
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

16) chain B
residue 363
type
sequence F
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

17) chain B
residue 364
type
sequence M
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

18) chain B
residue 449
type
sequence H
description BINDING SITE FOR RESIDUE 241 B 7001
source : AC2

19) chain B
residue 286
type BINDING
sequence Q
description BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
source Swiss-Prot : SWS_FT_FI1

20) chain B
residue 323
type BINDING
sequence H
description BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
source Swiss-Prot : SWS_FT_FI1

21) chain B
residue 449
type BINDING
sequence H
description BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
source Swiss-Prot : SWS_FT_FI1

22) chain B
residue 473
type BINDING
sequence Y
description BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
source Swiss-Prot : SWS_FT_FI1


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