eF-site ID 2j95-AB
PDB Code 2j95
Chain A, B

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Title CRYSTAL STRUCTURE OF A HUMAN FACTOR XA INHIBITOR COMPLEX
Classification HYDROLASE
Compound ACTIVATED FACTOR XA HEAVY CHAIN
Source ORGANISM_COMMON: HUMAN; ORGANISM_SCIENTIFIC: HOMO SAPIENS;
Sequence A:  IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTA
AHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRF
TKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLM
TQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSS
SFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVT
GIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT
B:  KLCSLDNGDCDQFCHEEQNSVVCSCARGYTLADNGKACIP
TGPYPCGKQTLE
Description


Functional site

1) chain A
residue 70
type
sequence D
description BINDING SITE FOR RESIDUE CA A1246
source : AC1

2) chain A
residue 72
type
sequence N
description BINDING SITE FOR RESIDUE CA A1246
source : AC1

3) chain A
residue 75
type
sequence Q
description BINDING SITE FOR RESIDUE CA A1246
source : AC1

4) chain A
residue 80
type
sequence E
description BINDING SITE FOR RESIDUE CA A1246
source : AC1

5) chain A
residue 96
type
sequence K
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

6) chain A
residue 97
type
sequence E
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

7) chain A
residue 98
type
sequence T
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

8) chain A
residue 99
type
sequence Y
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

9) chain A
residue 174
type
sequence F
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

10) chain A
residue 189
type
sequence D
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

11) chain A
residue 190
type
sequence A
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

12) chain A
residue 192
type
sequence Q
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

13) chain A
residue 195
type
sequence S
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

14) chain A
residue 213
type
sequence V
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

15) chain A
residue 215
type
sequence W
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

16) chain A
residue 216
type
sequence G
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

17) chain A
residue 219
type
sequence G
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

18) chain A
residue 226
type
sequence G
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

19) chain A
residue 227
type
sequence I
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

20) chain A
residue 228
type
sequence Y
description BINDING SITE FOR RESIDUE GSX A1245
source : AC2

21) chain B
residue 21-36
type prosite
sequence CSCARGYTLADNGKAC
description EGF_2 EGF-like domain signature 2. CtCleGFegkn....C
source prosite : PS01186

22) chain A
residue 53-58
type prosite
sequence LTAAHC
description TRYPSIN_HIS Serine proteases, trypsin family, histidine active site. LTAAHC
source prosite : PS00134

23) chain A
residue 189-200
type prosite
sequence DACQGDSGGPHV
description TRYPSIN_SER Serine proteases, trypsin family, serine active site. DAcqGDSGGPHV
source prosite : PS00135


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